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ʻO ka Tetracycline CAS: 60-54-8
He antibiotic ākea ka Tetracycline no ka papa tetracycline, i loaʻa mai ka hui kūlohelohe chlortetracycline. Hoʻopaʻa ia i ka hana protein bacteria ma o ka nakinaki ʻana i ka ribosome bacteria, a laila e pale ana i ka hoʻopili ʻana o ka aminoacyl-tRNA i ka hui mRNA-ribosome. ʻO kēia ʻano hana e alakaʻi ai i nā hopena bacteriostatic e kūʻē i kahi ākea o nā bacteria gram-positive a me gram-negative, a me kekahi mau protozoa.
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ʻO Teicoplanin CAS:61036-62-2
ʻO Teicoplanin kahi lāʻau antibiotic glycopeptide i loaʻa mai Actinoplanes teichomyceticus, kūpono i nā ʻano bacteria gram-positive like ʻole me ka methicillin-resistant Staphylococcus aureus (MRSA). Hoʻopaʻa ia i ka synthesis o ka paia cell bacteria ma o ka hoʻopaʻa ʻana i ka D-alanyl-D-alanine terminus o nā peptidoglycan precursors, e alakaʻi ana i ka lysis cell a me nā hopena bactericidal. Hoʻohana pinepine ʻia ʻo Teicoplanin i nā hoʻonohonoho lapaʻau no ka mālama ʻana i nā maʻi koʻikoʻi i hoʻokumu ʻia e nā meaola gram-positive.
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ʻO Sulfisoxazol (4-amino-N-(3,4-dimethyl-5-isoxazolyl)benzenesulfonamide) CAS:127-69-5
ʻO Sulfisoxazole, i ʻike ʻia hoʻi ʻo sulfafurazole, he antibiotic sulfonamide ia no ka papa lāʻau sulfa. Ua wehewehe ʻia me ke kemika he 4-amino-N-(3,4-dimethyl-5-isoxazolyl)benzenesulfonamide, kāohi ka sulfisoxazole i ka ulu ʻana o ka bacteria ma ke keakea ʻana i ka synthesis o ka folic acid. Kuhi kēia ʻano hana i ka dihydropteroate synthase, kahi enzyme koʻikoʻi no ka hana ʻana o ka folate bacteria, a laila e keakea ana i ko lākou ulu ʻana a me ka hoʻolaha ʻana.
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Sulfapyridine CAS:144-83-2
He lāʻau antibiotic sulfonamide ka Sulfapyridine i hoʻohana mua ʻia i ka mālama ʻana i nā maʻi bacteria, ʻoiai i ka wā o ke Kaua Honua II. No ka papa o nā lāʻau sulfa ia, kahi e kāohi ai i ka ulu ʻana o ka bacteria ma ke keakea ʻana i ka synthesis o ka waikawa folic. Hoʻopuka ka Sulfapyridine i kāna mau hopena bacteriostatic ma ka hoʻopaʻa ʻana i ka dihydropteroate synthase, kahi enzyme koʻikoʻi no ka hana folate i loko o ka bacteria.
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ʻO Tazobactam CAS:89786-04-9
He mea hoʻopale beta-lactamase ʻo Tazobactam e hoʻonui ai i ka hana o nā antibiotic beta-lactam ma ka pale ʻana iā lākou mai ka hoʻohaumia ʻia e nā enzyme beta-lactamase i hana ʻia e nā bacteria kūʻē he nui. Hoʻohana pinepine ʻia ia me nā antibiotic beta-lactam e like me piperacillin e hoʻonui i kā lākou hana e kūʻē i nā ʻano maʻi bacteria like ʻole. Hoʻihoʻi maikaʻi ʻo Tazobactam i ka pono o nā antibiotic beta-lactam e kūʻē i nā bacteria beta-lactamase-producing, ʻoiai nā meaola gram-negative.
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ʻO Tigecycline CAS:220620-09-7
He antibiotic glycylcycline ākea ka Tigecycline e kāohi ana i ka hana ʻana o ka protein bacteria ma o ka hoʻopaʻa ʻana i ka subunit ribosomal 30S, no laila e hoʻopuka ana i nā hopena bacteriostatic e kūʻē i nā ʻano bacteria gram-positive a me gram-negative, me nā pathogens multidrug-resistant. He pili ia i ke ʻano me nā tetracyclines akā loaʻa iā ia ka hana i hoʻonui ʻia e kūʻē i nā ʻano kūʻē ma muli o kona ʻano hana kūikawā a me nā hoʻololi ʻana i ke ʻano.
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Paʻakai paʻakai Sulbactam CAS: 69388-84-7
ʻO ka paʻakai sodium Sulbactam kahi mea hoʻopaʻa beta-lactamase i hoʻohana pinepine ʻia me kekahi mau antibiotics e hakakā i nā maʻi bacteria. Hana ia ma ke kāohi ʻana i ka hana o nā enzymes beta-lactamase i hana ʻia e ka bacteria, hiki ke hoʻolilo i nā antibiotics i mea ʻole. Ma ka pale ʻana i ka hōʻino ʻana o nā antibiotics e like me penicillins a me cephalosporins, kōkua ka paʻakai sodium sulbactam i ka hoʻonui ʻana i ko lākou mau waiwai antibacterial. Hoʻohana pinepine ʻia kēia hui me nā antibiotics e like me ampicillin e hana i nā hopena synergistic e kūʻē i nā ʻano bacteria like ʻole.
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Sulfadimidine CAS:57-68-1
ʻO Sulfadimidine, i ʻike ʻia hoʻi ʻo sulfamethazine, he antibiotic sulfonamide i hoʻohana ʻia i ka mālama ʻana i nā maʻi bacteria. No ka papa o nā antimicrobial i ʻike ʻia he mau lāʻau sulfa, e hana ana ma ke kāohi ʻana i ka ulu ʻana o ka bacteria a me ka hana hou ʻana. Hoʻopilikia ʻo Sulfadimidine i ka synthesis o ka folic acid i loko o ka bacteria, kahi ʻāpana koʻikoʻi no ko lākou ola ʻana, e alakaʻi ana i nā hopena bacteriostatic e kūʻē i kahi ākea o nā bacteria gram-positive a me gram-negative.
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Paʻakai sodium Sulfacetamide CAS: 6209-17-2
ʻO ka paʻakai sodium Sulfacetamide kahi mea i hoʻoheheʻe ʻia i ka wai o ka sulfacetamide, kahi antibiotic sulfonamide i hoʻohana pinepine ʻia i nā ʻano hana topical no ka mālama ʻana i nā maʻi bacteria o ka ʻili a me nā maka. Hoʻonui kēia ʻano paʻakai i ka solubility a me ke kūpaʻa o ka sulfacetamide, e kūpono ai no nā noi lāʻau lapaʻau like ʻole. Hana ka paʻakai sodium Sulfacetamide ma ke kāohi ʻana i ka ulu ʻana o nā bacteria, ʻoiai nā mea kuleana no nā kūlana e like me ka acne vulgaris, seborrheic dermatitis, a me nā maʻi maka e like me ka conjunctivitis. Hoʻopilikia ia i ka synthesis folate bacteria, e kuhikuhi pono ana i kahi ākea ākea o nā bacteria gram-positive a me gram-negative.
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ʻO ka Streptomycin sulfate CAS: 3810-74-0
He lāʻau antibiotic ʻo Streptomycin sulfate no ka papa aminoglycoside. Loaʻa ia mai ka bacteria Streptomyces griseus a hoʻohana pinepine ʻia e mālama i nā maʻi bacteria. Hana ʻo Streptomycin sulfate ma ke kāohi ʻana i ka hana ʻana o ka protein bacteria, a laila e pepehi pono ana i nā bacteria hiki ke maʻalahi. Hoʻomaopopo pinepine ʻia no ka mālama ʻana i ka maʻi puʻupuʻu, ka maʻi ahulau, ka tularemia, a me kekahi mau maʻi ʻē aʻe i hoʻokumu ʻia e nā bacteria hiki ke maʻalahi. Loaʻa pinepine ʻo Streptomycin sulfate ma ke ʻano injectable a lawelawe ʻia ma ke ʻano intramuscularly a i ʻole intravenously ma lalo o ka nānā ʻana o ke kauka.
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Paʻakai paʻakai Sulfamethoxazole CAS: 4563-84-2
ʻO ka paʻakai sodium Sulfamethoxazole kahi hopena wai-hoʻoheheʻe ʻia o ka sulfamethoxazole, kahi antibiotic sulfonamide i hoʻohana ʻia i ka mālama ʻana i nā maʻi bacteria. Hoʻonui kēia ʻano paʻakai i ka solubility a me ke kūpaʻa o ka sulfamethoxazole, e kūpono ai no nā ʻano lāʻau lapaʻau like ʻole. Hoʻopuka ka paʻakai sodium Sulfamethoxazole i kona hopena bacteriostatic ma ke kāohi ʻana i ka synthesis o ka waikawa folic i loko o ka bacteria, kahi hana koʻikoʻi no ko lākou ulu ʻana a me ka hana hou ʻana. He kūpono ia e kūʻē i kahi ākea o nā bacteria gram-positive a me gram-negative.
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Sulfamethoxazole CAS:723-46-6
ʻO Sulfamethoxazole kahi antibiotic sulfonamide i hoʻohana pinepine ʻia me ka trimethoprim e hana i kahi lāʻau antibacterial ikaika i ʻike ʻia ʻo co-trimoxazole a i ʻole trimethoprim-sulfamethoxazole (TMP-SMX). No ka papa o nā antimicrobial i ʻike ʻia ʻo nā lāʻau sulfa, ka mea e kāohi ai i ka ulu ʻana o ka bacteria ma ke keakea ʻana i ka synthesis o ka folic acid. Hoʻopilikia kūikawā ʻo Sulfamethoxazole i ka dihydropteroate synthase, kahi enzyme i komo i ka hana folate, no laila e hoʻopuka ana i nā hopena bacteriostatic e kūʻē i kahi ākea ākea o nā bacteria gram-positive a me gram-negative.
