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Venlafaxine CAS:93413-69-5

He lāʻau antidepressant ʻo Venlafaxine o ka papa serotonin a me norepinephrine reuptake inhibitor (SNRI). Ua hoʻomohala mua ʻia kēia lāʻau e Wyeth ma 19Chemicalbook93 a ke kūʻai ʻia aku nei e Pfizer. Ua ʻae ʻia kēia lāʻau no ka mālama ʻana i ka maʻi kaumaha nui (MDD), ka maʻi hopohopo maʻamau (GAD), a me ke kaumaha e pili ana me ka hopohopo.


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Hoʻohana a me ka hopena

Hiki iā Venlafaxine ke kāohi i ka reuptake o NA a me 5-HT, a kāohi iki hoʻi i ka reuptake o dopamine. In vitro inhibition of cholinergic receptors, histamine receptors α ʻAʻohe pilina o nā receptors ʻelua. Maikaʻi ka omo ʻana o ka Gastrointestinal, a ua metabolized ʻia ʻo Chemicalbook e cytochrome P45011D6 i loko o ke akepaʻa a hoʻokuʻu ʻia e ka mimi. ʻO ka t1/2 o nā metabolites hana nui mai 5 a 11 mau hola. Ma hope o 3 mau pule, ua hiki i ka paʻa o ke kūlana paʻa. Hoʻohana ʻia no ka mālama ʻana i ke kaumaha.

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ʻIke Hou Aʻe:

Hoʻonohonoho ʻana C17H27NO2
Hoʻāʻo 99%
helehelena Pauka aniani keʻokeʻo
Helu CAS. 93413-69-5
Hoʻopili ʻana 25KG
Ola Papa 2 mau makahiki
Ka Waihona E mālama i kahi maloʻo a me kahi anuanu
Palapala hōʻoia ISO.

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